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GSK2798745

Glpbio
Catalog No:GC39387-10mg CAS No.:1419609-94-1 MDLNo: Brand:Glpbio purity: 特性: Purpose:GSK2798745 是一流的,高效的,選擇性的且具有口服活性的 瞬時(shí)受體電位香草酸 4 (TRPV4) 離子通道阻斷劑,對(duì)于 hTRPV4 和 rTRPV4 的 IC50 值分別為 1.8 和 1.6 nM。GSK2798745 用于治療與充血性心力衰竭相關(guān)的肺水腫的研究。DMSO: 250 mg/mL (542.85 mM)
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