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Home > Category > > Small Molecule Compound > Balixafortide TFA

Balixafortide TFA

Glpbio
Catalog No:GC39343-25mg CAS No.: MDLNo: Brand:Glpbio purity: 特性: Purpose:Balixafortide TFA (POL6326 TFA) 是一種有效的,選擇性的,耐受性好的肽類 CXCR4 拮抗劑,其 IC50 小于 10 nM。Balixafortide TFA 對(duì) CXCR4 的選擇性比包括 CXCR7 在內(nèi)的許多受體高出 1000 倍。Balixafortide TFA 以 IC50 < 10 nM 阻斷 β-arrestin 募集和鈣通量。Balixafortide TFA 還是一種有效的造血干細(xì)胞和祖細(xì)胞 (HSPC) 動(dòng)員劑,并具有抗癌作用。Soluble in DMSO
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