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BRD5648

Glpbio
Catalog No:GC39263-10mg CAS No.:2056261-42-6 MDLNo: Brand:Glpbio purity: 特性: Purpose:BRD5648 ((R)-BRD0705) 是一種無活性的 BRD0705 的 R 型異構(gòu)體,BRD0705 是一種有效的,具有旁系選擇性和口服活性的 GSK3α 抑制劑,IC50 為 66 nM,Kd 為 4.8 μM。BRD0705 與 GSK3β (IC50 為 515 nM) 相比,對 GSK3α 的選擇性更高 (8 倍)。BRD0705 可用于急性髓細胞性白血病。DMSO: 300 mg/mL (933.36 mM)
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