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Home > Category > > Small Molecule Compound > LP-935509

LP-935509

Glpbio
Catalog No:GC39256-100mg CAS No.:1454555-29-3 MDLNo: Brand:Glpbio purity: 特性: Purpose:LP-935509 是一種小分子銜接蛋白-2 相關(guān)激酶1 (AAK1) 選擇性和腦滲透抑制劑 (IC50=3.3 nM),一種 ATP 競(jìng)爭(zhēng)性抑制劑,其 Ki 為 0.9 nM。 LP-935509 是 BIKE 的有效抑制劑 (IC50=14 nM) 和適度的 GAK 抑制劑 (IC50=320 nM)。 LP-935509 可逆轉(zhuǎn) SNL 手術(shù)后的疼痛。DMSO: 250 mg/mL (630.61 mM)
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