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Home > Category > > Small Molecule Compound > 1-Naphthohydroxamic acid

1-Naphthohydroxamic acid

Glpbio
Catalog No:GC39214-50mg CAS No.:6953-61-3 MDLNo: Brand:Glpbio purity: 特性: Purpose:1-Naphthohydroxamic acid (Compound 2) 是一種有效的,選擇性的 HDAC8 抑制劑,IC50 為 14 μM。1-Naphthohydroxamic acid 對 HDAC8 的選擇性高于 I 類 HDAC1 和 II 類 HDAC6 (IC50 100 μM)。1-Naphthohydroxamic acid 不會增加整體組蛋白 H4 的乙?;?,也不會降低總細(xì)胞內(nèi) HDAC 的活性。1-Naphthohydroxamic acid 可誘導(dǎo)微管蛋白乙?;?。DMSO: 125 mg/mL (667.77 mM)
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