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SR-4835

Glpbio
Catalog No:GC39175-100mg CAS No.:2387704-62-1 MDLNo: Brand:Glpbio purity: 特性: Purpose:SR-4835 是有效,高選擇性和 ATP 競爭性的 CDK12/CDK13 雙重抑制劑 (CDK12:IC50=99 nM,Kd=98 nM;CDK13:Kd=4.9 nM)。SR-4835 與破壞 DNA 的化學療法和 PARP 抑制劑協(xié)同作用,并引起三陰性乳腺癌 (TNBC) 細胞凋亡。DMSO: 5 mg/mL (10.01 mM; ultrasonic and warming and heat to 60°C)
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