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Home > Category > > Small Molecule Compound > Pozanicline dihydrochloride

Pozanicline dihydrochloride

Glpbio
Catalog No:GC38940-1mg CAS No.:161416-61-1 MDLNo: Brand:Glpbio purity: 特性: Purpose:Pozanicline dihydrochloride (ABT-089 dihydrochloride) 是一種具有口服活性的煙堿型乙酰膽堿受體 (nAChR) 激動劑,與 [3H] 胱氨酸位點(diǎn)結(jié)合,Ki 為 16.7 nM。Pozanicline dihydrochloride 是一種 α4β2 選擇性 nAChR 激動劑,與大鼠腦 α4β2 nAChR 結(jié)合,Ki 為 17 nM,而與 α7nAChR 的結(jié)合力很弱。Soluble in DMSO
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