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Home > Category > > Small Molecule Compound > TRAF-STOP inhibitor 6877002

TRAF-STOP inhibitor 6877002

Glpbio
Catalog No:GC38868-10mg CAS No.:433249-94-6 MDLNo: Brand:Glpbio purity: 特性: Purpose:TRAF-STOP inhibitor 6877002,一種抑制 CD40-TRAF6 相互作用的選擇性抑制劑,從專利 WO2014033122A1 中獲得,抑制 RAW 細胞中 NF-κB 活化,化合物VII。TRAF-STOP 6877002 可阻止小鼠中已發(fā)生的動脈粥樣硬化惡化,減少白細胞募集并減少巨噬細胞活化;減少動脈粥樣硬化斑塊中的巨噬細胞增殖。DMSO: 125 mg/mL (497.37 mM)
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