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TBOPP

Glpbio
Catalog No:GC38855-5mg CAS No.:1996629-79-8 MDLNo: Brand:Glpbio purity: 特性: Purpose:TBOPP 是一種 DOCK1 的選擇性抑制劑,其 IC50 為 8.4 μM。TBOPP 以高親和力 (Kd 為 7.1 μM) 與 DOCK1 DHR-2 結(jié)構(gòu)域結(jié)合,對(duì)廣泛類(lèi)型的腫瘤均具有抗腫瘤活性。DMSO: 125 mg/mL (254.85 mM)
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