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Lapaquistat acetate

Glpbio
Catalog No:GC38807-1mg CAS No.:189060-13-7 MDLNo: Brand:Glpbio purity: 特性: Purpose:Lapaquistat acetate (TAK-475) 是一種角鯊烯合酶 (squalene synthase) 抑制劑,可阻止法呢基二磷酸酯 (FPP) 轉(zhuǎn)化為角鯊烯。Lapaquistat acetate (TAK-475) 最初旨在用于甲羥戊酸激酶缺乏癥 (MKD),可有效降低低密度脂蛋白膽固醇,但可能引起肝臟損害。DMSO: 46 mg/mL (71.30 mM)
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