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Home > Category > > Small Molecule Compound > CKI-7

CKI-7

Glpbio
Catalog No:GC38755-5mg CAS No.:120615-25-0 MDLNo: Brand:Glpbio purity: 特性: Purpose:CKI-7 是一種有效且 ATP 競爭性的酪蛋白激酶 1 (CK1) 抑制劑,IC50 為 6 μM,Ki 為 8.5 μM。CKI-7 選擇性抑制 Cdc7 激酶,還抑制 SGK,S6K1 以及 MSK1。CKI-7 對(duì)酪蛋白激酶 II 和其他蛋白激酶的作用弱得多。DMSO: 25 mg/mL (87.49 mM)
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