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Home > Category > > Small Molecule Compound > TVB-3166

TVB-3166

Glpbio
Catalog No:GC38710-10mg CAS No.:1533438-83-3 MDLNo: Brand:Glpbio purity: 特性: Purpose:TVB-3166 是一種口服有效,可逆和選擇性脂肪酸合成酶 (FASN) 抑制劑,對(duì)于 FASN 和細(xì)胞棕櫚酸酯合成的 IC50 分別為 42 nM 和 81 nM。TVB-3166 誘導(dǎo)細(xì)胞凋亡,并抑制體內(nèi)異種移植腫瘤的生長(zhǎng)。DMSO: 62.5 mg/mL (162.56 mM)
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