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Home > Category > > Small Molecule Compound > PXS-5153A monohydrochloride

PXS-5153A monohydrochloride

Glpbio
Catalog No:GC38583-1mg CAS No.: MDLNo: Brand:Glpbio purity: 特性: Purpose:PXS-5153A monohydrochloride 是一種有效的、選擇性的、具有口服活性和快速起效的賴氨酰氧化酶 2/3 (LOXL2/LOXL3) 的雙抑制劑,對幾乎所有哺乳動物L(fēng)OXL2的IC50 均< 40 nM,對人類LOXL3 的IC50 為63 nM。PXS-5153A monohydrochloride 可減少交聯(lián),改善纖維化。DMSO: 250 mg/mL (569.54 mM)
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