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ATI-2341 TFA

Glpbio
Catalog No:GC38541-10mg CAS No.: MDLNo: Brand:Glpbio purity: 特性: Purpose:ATI-2341 是一種有效的 C-X-C 趨化因子受體 4 型 (CXCR4) 功能選擇性變構(gòu)激動(dòng)劑,其作為偏向配體起作用,有利于 Gα1激活而不是 Gα13。ATI-2341 激活抑制性異源三聚體 G 蛋白 (Gi) 以促進(jìn) cAMP 產(chǎn)生的抑制并誘導(dǎo)鈣動(dòng)員。ATI-2341 是一種有效骨髓多形核中性粒細(xì)胞 (PMNs) 和造血干細(xì)胞和祖細(xì)胞 (HSPCs) 動(dòng)員劑。DMSO: 100 mg/mL (42.18 mM)
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