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C-178

Glpbio
Catalog No:GC38494-5mg CAS No.:329198-87-0 MDLNo: Brand:Glpbio purity: 特性: Purpose:C-178,STING 的共價抑制劑,與 Cys91 有效結合并選擇性地抑制小鼠中不同的激活劑引起的 STING 反應。C-178 選擇性地降低 STING- 而非 RIG-I- 或 TBK1- 介導的 IFN-β 報告基因活性。C-178 阻斷棕櫚?;?(PMA) 誘導的 STING 類聚;抑制 CMA 誘導的 TBK1 (STING 下游蛋白激酶) 磷酸化。DMSO: 41.67 mg/mL (129.30 mM)
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