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Home > Category > > Small Molecule Compound > BMS-986020 sodium

BMS-986020 sodium

Glpbio
Catalog No:GC38470-50mg CAS No.:1380650-53-2 MDLNo: Brand:Glpbio purity: 特性: Purpose:BMS-986020 sodium 是高親和力溶血磷脂酸受體 1 (LPA1) 拮抗劑。BMS-986020 sodium 抑制膽汁酸和磷脂轉運蛋白,抑制 BSEP,MRP4 和 MDR3,IC50 值分別為 4.8 μM,6.2 μM 和 7.5 μM。BMS-986020 sodium 用于治療特發(fā)性肺纖維化 (IPF)。DMSO: 150 mg/mL (297.32 mM); H2O: < 0.1 mg/mL (insoluble)
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