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WRG-28

Glpbio
Catalog No:GC38206-50mg CAS No.:1913291-02-7 MDLNo: Brand:Glpbio purity: 特性: Purpose:WRG-28 是選擇性,細(xì)胞外作用的 DDR2 變構(gòu)抑制劑,IC50 為 230 nM。WRG-28 通過受體的變構(gòu)調(diào)節(jié)特異地抑制受體-配體相互作用。WRG-28 通過靶向 DDR2 抑制腫瘤侵襲和遷移,基質(zhì)的腫瘤支持作用,并抑制肺中的轉(zhuǎn)移性乳腺腫瘤細(xì)胞定植。DMSO: 15.62 mg/mL (38.06 mM)
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