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Home > Category > > Small Molecule Compound > Raphin1

Raphin1

Glpbio
Catalog No:GC38189-25mg CAS No.:2022961-17-5 MDLNo: Brand:Glpbio purity: 特性: Purpose:Raphin1 是一種口服生物可利用的,選擇性調節(jié)性磷酸酶 PPP1R15B (R15B) 抑制劑。Raphin1 與 R15B-PP1c 全磷酸酶強烈結合 (Kd=33 nM),與 R15A-PP1c 相比,結合 R15B-PP1c 約為其 30 倍的選擇性。Raphin1 穿過血腦屏障,并減少蛋白質錯誤折疊疾病的小鼠模型中的生物和分子缺陷。DMSO: 125 mg/mL (540.94 mM)
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