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Home > Category > > Small Molecule Compound > ML753286

ML753286

Glpbio
Catalog No:GC38129-5mg CAS No.:1699720-89-2 MDLNo: Brand:Glpbio purity: 特性: Purpose:ML753286 是一種口服活性和選擇性 BCRP (抗乳腺癌蛋白) 抑制劑,IC50 為 0.6 μM。 ML753286 在嚙齒動物和人類肝臟 S9 組分中具有高滲透性和低至中等清除率,并且在不同物種中都具有血漿穩(wěn)定性。Soluble in DMSO
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