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Home > Category > > Small Molecule Compound > (R)-VU 6008667

(R)-VU 6008667

Glpbio
Catalog No:GC38110-25mg CAS No.:2097818-14-7 MDLNo: Brand:Glpbio purity: 特性: Purpose:(R)-VU6008667 是 VU6008667 的活性對(duì)映異構(gòu)體,是一種口服活性的乙酰膽堿受體 5 亞型 (M5 NAM) 抑制劑,IC50 值分別為 1.2 μM (human) 和 1.6 μM (rat)。(R)-VU6008667 對(duì) M5 的選擇性高于 M1-4,CNS 滲透率高。DMSO: 100 mg/mL (227.87 mM)
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