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TH5487

Glpbio
Catalog No:GC37776-100mg CAS No.:2304947-71-3 MDLNo: Brand:Glpbio purity: 特性: Purpose:TH5487 是一種有效的 8-氧鳥嘌呤 DNA 糖基化酶1 (OGG1) 抑制劑,IC50 為342 nM,TH5487 阻止 OGG1 識(shí)別其 DNA 底物,抑制 DNA 修復(fù)和修飾 OGG1 染色質(zhì)動(dòng)力學(xué),從而抑制促炎基因。DMSO: 25 mg/mL (46.20 mM)
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